Definition of AntiandrogenAntiandrogen: A drug that blocks the action of androgens (male sex hormones). Antiandrogens are sometimes used in the treatment of prostate cancer. The antiandrogens currently available include flutamide (Eulexin), bicalutamide (Casodex), and nilutamide (Nilandron). Source: MedTerms™ Medical Dictionaryhttp://www.medterms.com/script/main/art.asp?articlekey=9824 Last Editorial Review: 6/14/2012
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